20
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T40999 | NMDA receptor antagonist 2 | ||
NMDA receptor antagonist 2 is a highly potent and orally active NR2B subtype-selective antagonist of the N-methyl-D-aspartate (NMDA) receptor. It exhibits remarkable binding affinities, with an IC50 of 1.0 nM and a Ki va... | |||
T60792 | NMDA receptor antagonist-3 | ||
NMDA receptor antagonist-3 is a NMDA receptor antagonist with a significan recovery rate (40.0%, at 100 μM) and safe toxicological characteristics in SH-SY5Y and human adipose mesenchymal stem cells. | |||
T79374 | NMDA receptor antagonist 7 | iGluR | |
Compound (S)-10a, a GluN2B subunit-selective NMDA receptor antagonist, exhibits a K i of 93 nM and an IC 50 of 72 nM. It is potentially useful for research into neurodegenerative diseases [1]. | |||
T79375 | NMDA receptor antagonist 8 | iGluR | |
Compound (R)-10a, an NMDA receptor antagonist, exhibits selectivity for the GluN2B subunit, possessing a Ki of 265 nM and an IC50 of 62 nM. This compound is utilized in research pertaining to neurodegenerative diseases [... | |||
T61924 | NMDA receptor modulator 6 | ||
NMDA receptor regulator 6 (Compound 183) is an effective NMDA receptor regulator and has research value in neurological disorders. | |||
T63003 | NMDA receptor potentiator-1 | ||
NMDA receptor potentiator-1 (Compound 1368) is a subunit-selective NMDA receptor enhancer with IC50 values of 4 μM and 5 μM for NR2C and NR2D expression, respectively. | |||
T61470 | NMDA receptor antagonist 5 | ||
NMDA receptor antagonist 5 (Compound 10e), a potent and non-toxic NMDA receptor antagonist, exhibits brain permeability. It is of significance in studying neurological disorders [1]. | |||
T60685 | NMDA receptor modulator 3 | ||
NMDA receptor modulator 3 (Compound 99) is a potent modulator of NMDA receptor that can be used in the research of neurological disorder [1]. | |||
T79273 | NMDA receptor antagonist 6 | iGluR | |
NMDA Receptor Antagonist 6 (Compound 13b) functions as an antagonist at the glycine-binding site of the NMDA receptor and demonstrates cytoneuroprotective efficacy. It safeguards PC12 cells from NMDA-induced damage and a... | |||
T61117 | NMDA receptor modulator 5 | ||
NMDA receptor modulator 5 (Compound 195), a potent NMDA receptor modulator, exhibits potential for neurological disorder research [1]. | |||
T60552 | NMDA receptor modulator 2 | ||
NMDA receptor modulator 2 (Compound 1) is a potent modulator of the NMDA receptor that can be used for neurological disorder research [1]. | |||
T60960 | NMDA receptor modulator 4 | ||
NMDA receptor modulator 4 (Compound 169) can be used for the research of neurological disorder that is a potent modulator of NMDA receptor [1]. | |||
T60306 | NMDA receptor antagonist 4 | ||
NMDA receptor antagonist 4 (IIc) is an uncompetitive, voltage-dependent, orally active NMDAR blocker, with an IC 50 of 1.93 μM. NMDA receptor antagonist 4 shows a positive predicted blood-brain-barrier (BBB) permeability... | |||
T4979 | Procyclidine hydrochloride | (±)-Procyclidine hydrochlorid | NMDAR , iGluR |
Procyclidine hydrochloride ((±)-Procyclidine hydrochlorid) is a potent anticholinergic agent and also have NMDA antagonist properties. | |||
T9157 | GP130 receptor agonist-1 | N-(4-Fluorophenyl)-4-phenyl-2-thiazolami | Interleukin |
GP130 receptor agonist-1 (N-(4-Fluorophenyl)-4-phenyl-2-thiazolami) is a potent, brain-penetrant and orally active GP130 receptor agonist. | |||
T6134 | IEM 1754 2HBr | IEM 1754 dihydrobromide | GluR |
IEM 1754 2HBr (IEM 1754 dihydrobromide) is a selective AMPA/kainate receptor blockers for GluR1 and GluR3 with IC50 of 6 μM. | |||
T16286 | Nelonemdaz | Neu2000 | Topoisomerase |
Neu2000 is an uncompetitive antagonist of N-methyl-D-aspartate (NMDA) receptor. | |||
T23449 | TCS 46b | NMDAR | |
NR1A/NR2B NMDA receptor antagonist,orally active | |||
T1186L | Ifenprodil | RC 61-91,RC-61-91,RC61-91,RC 6191 | Adrenergic Receptor , NMDAR |
Ifenprodil (RC61-91) is an inhibitor of the NMDA receptor, specifically of GluN1 (glycine-binding NMDA receptor subunit 1) and GluN2B (glutamate-binding NMDA receptor subunit 2) subunits. Additionally, Ifenprodil inhibit... | |||
T27178 | Dimiracetam | ISF4185,ISF-4185,NT11624,NT-11624,BND11624,BND-11624 | |
Dimiracetam, a NMDA-receptor antagonist, is used potentially for the treatment of neuropathic pain. |